专利名称 | Radiolabelled octreotate analogues as PET tracers | ||
申请号 | US14002168 | 申请日 | |
公开(公告)号 | US10201625B2 | 公开(公告)日 | 2012-03-01 |
申请(专利权)人 | 发明人 | Sajinker Kaur Luthra; Julius Leyton; Eric Ofori Aboagye; Lisa Iddon; Bard Indrevoll; Matthias Eberhard Glaser; Alan Cuthbertson | |
专利来源 | 国家知识产权局 | 转化方式 | |
摘要 |
Novel radiotracer(s) for Positron Emission Tomography (PET) imaging are described. Novel radiotracer(s) for Positron Emission Tomography (PET) imaging of neuorendocrine tumors are described. Specifically the present invention describes novel [18F]Fluoroethyltriazol-[Tyr3]Octreotate analogs; in particular those that target somatostatin receptors found on the cell surface of gastroenteropancreatic neuorendocrine tumors. The present invention also describes intermediate(s), precursor(s), pharmaceutical composition(s), methods of making, and methods of use of the novel radiotracer(s). |