专利名称 | PREPARATION METHOD FOR FUSED TRICYCLIC γ-AMINO ACID DERIVATIVE AND INTERMEDIATE THEREOF | ||
申请号 | WOCN19096522 | 申请日 | |
公开(公告)号 | WO2020029762A1 | 公开(公告)日 | |
申请(专利权)人 | SICHUAN HAISCO PHARMACEUTICAL CO LTD | 发明人 | FAN Jiang; CHEN Qingping; WANG Chengtao; FENG Jianchuan |
专利来源 | 国家知识产权局 | 转化方式 | |
摘要 |
A preparation method for a fused tricyclic γ-amino acid derivative and an intermediate thereof, and a method for preparing an intermediate of the fused tricyclic γ-amino acid derivative. The fused tricyclic γ-amino acid derivative has a structure as represented by formula (I). The preparation method uses readily available raw materials and comprises simple steps; the entire synthesis process uses crystallization purification, while silica gel column chromatography or other preparatory chromatography methods are not used, being suitable for large-scale industrial production. |